OnCo
drugsProductNot mapped hereapproved

Imetelstat

Imetelstat is the first telomerase-blocking drug approved for any cancer; it frees many lower-risk MDS patients from transfusions after growth factors have failed.

IMerge (NEJM 2024): 8-week transfusion independence 40% vs 15% with placebo, with durable responses and reductions in mutant allele burden suggesting disease modification. Cytopenias are the main toxicity. Phase 3 in JAK-inhibitor-refractory myelofibrosis (IMpactMF) tests overall survival.

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Imetelstat (thio-phosphoramidate oligonucleotide) · 2D coordinates (no PubChem conformer)
PubChem
Modality
Telomerase inhibitor (oligonucleotide)
Mechanism
13-mer lipid-conjugated oligonucleotide that binds the RNA template of telomerase (hTR), inhibiting telomerase in malignant clones with high telomerase activity.
Brand / code
Rytelo
Medicare
Part B (clinician-administered)

Given by infusion or injection in a clinic or hospital outpatient department, so it is a Part B drug: Medicare pays 80% after the Part B deductible and the patient owes 20% coinsurance, uncapped in Original Medicare unless a Medigap policy applies. Every-four-week infusion for lower-risk MDS (approved June 2024).

Commercial insurance
covered with prior authorisation

Covered under the medical benefit with prior authorisation confirming diagnosis, biomarker status and line of therapy; site-of-care policies may steer infusions away from hospital outpatient departments. Transfusion-dependent lower-risk MDS after ESA failure.

20% Part B coinsurance on a high-cost infusion adds up quickly: Medigap Plan G or N, Medicare Advantage maximum out-of-pocket, Medicaid dual eligibility, or a charity fund are the usual buffers.

Sources: Medicare.gov: Chemotherapy · Medicare.gov: Prescription drugs (outpatient, Part B). Not medical or financial advice; verify with your plan.

Not yet researchedSearch NICE
Notes
EU-licensed 2025 for lower-risk MDS anaemia; UK licence and NICE position not yet researched.

Sources: NICE search: imetelstat. Funding decisions are indication-specific and change monthly; verify with NICE and your treating team.

Regulatory

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Approvals

RegionYearIndication
US2024Low- to intermediate-1-risk MDS with transfusion-dependent anaemia after ESA failure
EU2025Lower-risk MDS transfusion-dependent anaemia

Trials

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Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
Imetelstat
intervention: Imetelstat
Open on ClinicalTrials.gov →

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Key papers

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Latest papers

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Latest papers · live from Europe PMC
Open in Europe PMC

Query for this drug: (TITLE:"Imetelstat" OR ABSTRACT:"Imetelstat" OR TITLE:"Rytelo" OR ABSTRACT:"Rytelo") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about Imetelstat, not a curated reading list.

Connected

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