OnCo

FOLFIRI

Checked 2026-09-09

Metastatic colorectal first or second line (with bevacizumab, aflibercept, ramucirumab or an anti-EGFR antibody)

One cycle

every 14 days
1234567891011121314Irinotecan: 180 mg/m², IntravenousIrinotecanLeucovorin (folinic acid): 400 mg/m², IntravenousLeucovorin (folinic aci…Fluorouracil bolus: 400 mg/m², IntravenousFluorouracil bolusFluorouracil infusion: 2,400 mg/m², IntravenousFluorouracil infusion
14-day cycle, until progressionIntravenous Continuous infusion

Components

DrugDoseRouteDays
Irinotecan
Topoisomerase I inhibitor (camptothecin prodrug)
180 mg/m²IVD1
Leucovorin (folinic acid)
400 mg/m²IVD1
Fluorouracil bolus
Fluoropyrimidine antimetabolite
400 mg/m²IVD1
Fluorouracil infusion
Fluoropyrimidine antimetabolite
2,400 mg/m²IVD1, 2 (46 h infusion)
Cycles
until progression
14-day cycle
Emetogenicity
Moderate (30-90%)
G-CSF
Not routine

Notes

  • UGT1A1*28 homozygotes have higher neutropenia risk; consider a lower irinotecan start dose.

Used in

Source

NCCN Colon Cancer; Douillard, Lancet 2000

Reference doses for a typical adult from the cited protocol or label. Doses are adjusted for renal and hepatic function, age, performance status and prior toxicity, and institutional protocols vary. Verify against the current label and your local protocol before treating. Not medical advice.

Other regimens for these cancers