OnCo
drugsProductNot mapped hereapproved

Fluciclovine F-18

Fluciclovine F-18 was the first PET tracer approved for finding recurrent prostate cancer after treatment (2016), and has been largely superseded since 2020 by PSMA PET.

Approved May 2016 for suspected recurrence with rising PSA; detection ~68% overall, lower at low PSA. EMSPOT/EMPIRE-1 (Lancet 2021) showed fluciclovine-guided salvage radiotherapy improved failure-free survival. PSMA PET (Ga-68 PSMA-11, piflufolastat, flotufolastat) has higher detection and displaced it.

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Fluciclovine
PubChem
Modality
PET radiotracer (synthetic amino acid)
Mechanism
18F-labelled leucine analogue taken up via LAT1/ASCT2 amino-acid transporters upregulated in prostate cancer; low urinary excretion improves pelvic imaging.
Brand / code
Axumin
Medicare
Part B (clinician-administered)

Diagnostic radiopharmaceutical billed with the PET/CT scan under Part B for suspected prostate cancer recurrence; PSMA agents have largely displaced it.

Commercial insurance
variable

Covered by many plans for biochemical recurrence, but some now require PSMA PET as the preferred tracer.

Sources: Medicare.gov: Chemotherapy · Medicare.gov: Prescription drugs (outpatient, Part B) · Medicare.gov: Diagnostic non-laboratory tests (imaging). Not medical or financial advice; verify with your plan.

Not appraisedSearch NICE
Notes
EU-licensed but not commissioned for routine NHS use; PSMA PET is preferred.
NHS England
Not routinely funded

Sources: NICE search: fluciclovine F-18. Funding decisions are indication-specific and change monthly; verify with NICE and your treating team.

Regulatory

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Approvals

RegionYearIndication
US2016PET imaging in men with suspected prostate cancer recurrence based on elevated PSA
EU2017Same

Trials

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Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
Fluciclovine F-18
intervention: Fluciclovine F-18
Open on ClinicalTrials.gov →

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Latest papers

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Latest papers · live from Europe PMC
Open in Europe PMC

Query for this drug: (TITLE:"Fluciclovine F-18" OR ABSTRACT:"Fluciclovine F-18" OR TITLE:"Axumin" OR ABSTRACT:"Axumin") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about Fluciclovine F-18, not a curated reading list.

Connected

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