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Chemistry42 and Pharma.AI (Insilico)

Generative chemistry platform behind the first AI-discovered drug to reach phase 2, plus oncology candidates.

Insilico's rentosertib (TNIK, IPF) reported phase 2a results in 2025; oncology programmes include ISM3091 (USP1, licensed to Exelixis) and ISM5411.

Generic schematic · not to scale · placeholder for the drug discovery front
Guide RNA library · Knockout → dependency

How it works

Generative models for target discovery, molecule generation and trial outcome prediction.

Strengths
  • Clinical-stage validation of the platform
Limitations
  • Oncology assets early
Since
2020

Latest papers

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Latest papers · live from Europe PMC
Open in Europe PMC

Query for this technology: (TITLE:"Chemistry42 and Pharma.AI" OR ABSTRACT:"Chemistry42 and Pharma.AI" OR TITLE:"Insilico" OR ABSTRACT:"Insilico") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about Chemistry42 and Pharma.AI (Insilico), not a curated reading list.

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