OnCo
drugsProductApproved2026🇨🇳

Sonrotoclax

Sonrotoclax is a more potent, shorter-acting successor to venetoclax. It was approved for mantle cell lymphoma in May 2026 and is in late-stage trials with zanubrutinib for CLL.

Approved in China (late 2025) for relapsed MCL and CLL/SLL after BTK inhibitor, and in the US on 13 May 2026 (accelerated) for relapsed/refractory MCL after ≥2 lines including a BTK inhibitor (BGB-11417-201: ORR 52%, median DOR 15.8 months). In treatment-naive CLL, sonrotoclax + zanubrutinib (BGB-11417-101) produced uMRD in nearly all patients by 96 weeks; phase 3 CELESTIAL-TNCLL (vs venetoclax-obinutuzumab) completes 2026. Shorter half-life allows faster ramp-up and less overlapping myelosuppression.

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Sonrotoclax · 2D coordinates (no PubChem conformer)
PubChem
Mechanism, step by step
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1.Sonrotoclax occupies the BH3 groove of BCL-2

Modality
Small-molecule BCL-2 inhibitor (second generation)
Mechanism
Selective BH3-mimetic BCL-2 inhibitor with higher potency and shorter half-life than venetoclax; active against venetoclax-resistant G101V BCL2 in preclinical models.
Brand / code
Beqalzi · BGB-11417
Dosing & schedule
Route
Oral
Schedule
4-week ramp-up then 320 mg once daily until progression (MCL label); CLL trials use 160-320 mg with zanubrutinib lead-in
Monitoring
TLS during ramp-up, neutropenia, infections

Source: www.fda.gov/drugs/resources-information-approved-drugs/fda-grants-accelerated-approval-sonrotoclax-relapsed-or-refractory-mantle-cell-lymphoma. Doses are for orientation; the current label governs.

Not appraisedSearch NICE
Notes
No UK marketing authorisation as of September 2026, so no NICE appraisal. Access only through a clinical trial or a company early access scheme.
NHS England
Not routinely funded

Sources: NICE search: sonrotoclax. Funding decisions are indication-specific and change monthly; verify with NICE and your treating team.

Regulatory

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  1. 13 May 2026ApprovalUS

    Accelerated approval in MCL; priority review, Project Orbis source

Approvals

RegionYearIndication
China2025Relapsed/refractory MCL and CLL/SLL after BTK inhibitor
US2026Relapsed/refractory mantle cell lymphoma after ≥2 lines including a BTK inhibitor (accelerated)

Safety

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Toxicity profile
Adverse event
Neutropenia
Most common grade ≥3 event in MCL and CLL studies
Tumour lysis syndrome
Mitigated by 4-week ramp
Diarrhoea, nausea
Mostly low grade

Rates read from the source. Blank cells mean the figure was not sourced, not that it is zero.

Trials

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ClinicalTrials.gov · phase 2/3
refreshed 2026-09-09
36 studies17 recruiting31 Phase 25 Phase 3
Search “Sonrotoclax” on ClinicalTrials.gov →
Counts are from a name search and may include unrelated studies; up to 100 studies are summarised.

Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
Sonrotoclax
intervention: Sonrotoclax
Open on ClinicalTrials.gov →

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Landmark trials in OnCo

Latest papers

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Literature trend13 papers in the last 12 months+44% vs prior 12How this is computed
Latest papers · live from Europe PMC
Open in Europe PMC

Query for this drug: (TITLE:"Sonrotoclax" OR ABSTRACT:"Sonrotoclax" OR TITLE:"Beqalzi" OR ABSTRACT:"Beqalzi" OR TITLE:"BGB-11417" OR ABSTRACT:"BGB-11417") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about Sonrotoclax, not a curated reading list.

Connected

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