OnCo
drugsProductNegative

Tiragolumab

An immune-brake blocker that looked excellent in a phase 2 lung cancer trial and then failed every phase 3.

CITYSCAPE (phase 2, 2020) showed tiragolumab plus atezolizumab roughly doubled response rate in PD-L1-high NSCLC. Phase 3 SKYSCRAPER-01 (PD-L1-high NSCLC) missed PFS and OS; SKYSCRAPER-02 (extensive-stage SCLC) was negative; SKYSCRAPER-06 (non-squamous NSCLC) was worse than control. Roche discontinued most of the programme in 2024–25. Other anti-TIGIT antibodies (domvanalimab, ociperlimab) showed no clearer benefit.

Lesson: a small randomised phase 2 with a surrogate endpoint in a selected population can mislead; redundancy between checkpoints means blocking a second one does not necessarily add to PD-1/PD-L1 blockade.

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Tiragolumab bound to TIGIT (PDB 8JEO), backbone trace
RCSB PDB
How it works, step by step · animated schematic, not to scale
Immune checkpoint inhibitors
Modality
Monoclonal antibody (anti-TIGIT)
Mechanism
IgG1 anti-TIGIT with intact Fc; blocks TIGIT–PVR interaction on T and NK cells.
Brand / code
RG6058, MTIG7192A

Trials

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Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
Tiragolumab
intervention: Tiragolumab
Open on ClinicalTrials.gov →

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Latest papers

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Literature trend22 papers in the last 12 months+83% vs prior 12How this is computed
Latest papers · live from Europe PMC
Open in Europe PMC

Query for this drug: (TITLE:"Tiragolumab" OR ABSTRACT:"Tiragolumab" OR TITLE:"RG6058" OR ABSTRACT:"RG6058" OR TITLE:"MTIG7192A" OR ABSTRACT:"MTIG7192A") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about Tiragolumab, not a curated reading list.

Connected

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