OnCo
drugsProductPhase 3

Raludotatug deruxtecan

Raludotatug deruxtecan is a CDH6 ADC in phase 3 for platinum-resistant ovarian cancer.

Phase 1 ORR ~46% in heavily pretreated ovarian cancer; REJOICE-Ovarian01 phase 2/3 versus chemotherapy. Daiichi Sankyo/Merck.

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Payload: deruxtecan (linker + DXd) · 2D coordinates (no PubChem conformer)
PubChem
How it works, step by step · animated schematic, not to scale
Antibody-drug conjugate (ADC)
Mechanism, step by step
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1.Antibody binds CDH6 on the tumour cell surface

Modality
ADC
Mechanism
Anti-CDH6 IgG1 with DXd.
Brand / code
R-DXd, DS-6000
Payload
DXd
Linker
GGFG cleavable
Dosing & schedule
Route
IV infusion
Schedule
5.6 mg/kg every 3 weeks (phase 2/3 dose)
Monitoring
ILD, blood counts

Source: clinicaltrials.gov/study/NCT06161025. Doses are for orientation; the current label governs.

Regulatory

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  1. Oct 2024Filing / dealUS

    Merck co-development of R-DXd under the Daiichi Sankyo alliance source

Safety

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Toxicity profile
Adverse event
Nausea
Fatigue
Neutropenia
Anaemia

Events listed without rates were not read from a primary source; see the label. Blank cells mean the figure was not sourced, not that it is zero.

Cost & access

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Cost & access
CountryReimbursement
United StatesInvestigational (REJOICE-Ovarian01)

List prices are manufacturer or Medicare figures where publicly disclosed; net prices after rebates are usually lower. Reimbursement changes; check the payer.

Trials

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ClinicalTrials.gov · phase 2/3
refreshed 2026-09-09
9 studies4 recruiting6 Phase 24 Phase 3
Search “Raludotatug deruxtecan” on ClinicalTrials.gov →
Counts are from a name search and may include unrelated studies; up to 100 studies are summarised.

Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
Raludotatug deruxtecan
intervention: Raludotatug deruxtecan
Open on ClinicalTrials.gov →

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Latest papers

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Literature trend2 papers in the last 12 monthsHow this is computed
Latest papers · live from Europe PMC
Open in Europe PMC

Query for this drug: (TITLE:"Raludotatug deruxtecan" OR ABSTRACT:"Raludotatug deruxtecan" OR TITLE:"R-DXd" OR ABSTRACT:"R-DXd" OR TITLE:"DS-6000" OR ABSTRACT:"DS-6000") AND (cancer OR tumor OR tumour OR oncology OR carcinoma OR lymphoma OR leukemia OR leukaemia OR myeloma OR sarcoma OR melanoma OR glioma). Results are unfiltered search hits about Raludotatug deruxtecan, not a curated reading list.

Connected

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