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Acute myeloid leukaemia

Acute myeloid leukaemia is an aggressive blood cancer where, after 40 years of the same chemotherapy, a wave of targeted drugs (FLT3, IDH, BCL-2, menin) arrived.

Acute myeloid leukaemia is a cancer of immature myeloid cells that floods the marrow and blood within weeks. It is defined molecularly: WHO 2022 and ICC 2022 classify by driver genetics, and ELN 2022 assigns favourable, intermediate, or adverse risk from NPM1, CEBPA, core-binding-factor fusions, FLT3, TP53, KMT2A, and myelodysplasia-related mutations. Median age at diagnosis is 68, and outcomes diverge sharply by age and fitness.

Treatment split into two paradigms. Fit patients receive intensive 7+3 induction (unchanged since 1973) with a targeted add-on chosen by genetics: midostaurin or quizartinib for FLT3, gemtuzumab ozogamicin for CD33+ favourable and intermediate risk, CPX-351 for secondary AML, then high-dose cytarabine consolidation and allogeneic transplant for adverse or MRD-positive disease. Unfit patients, once offered only supportive care, now receive venetoclax with azacitidine (VIALE-A) or, since May 2026, an all-oral regimen with decitabine-cedazuridine; IDH1-mutated patients may receive ivosidenib-azacitidine (AGILE). Relapse is treated by genotype: gilteritinib (FLT3), ivosidenib, olutasidenib or enasidenib (IDH), and the new menin inhibitors revumenib and ziftomenib (NPM1-mutated or KMT2A-rearranged), with transplant as the consolidating cure.

Measurable residual disease by flow cytometry, NPM1 qPCR, or error-corrected NGS now decides transplant and maintenance, and platform trials such as myeloMATCH assign therapy from rapid genomics at diagnosis. The unsolved problems are TP53-mutated and complex-karyotype AML, where every new class has failed so far, relapse after transplant, early death from infection in older patients, and the cost and logistics of the increasingly individualised pathway.

State of the art today

  • Menin inhibitors.
  • Venetoclax combinations.
  • Genotype-directed induction: FLT3 inhibitors (two positive phase 3 trials), gemtuzumab for CD33+ favourable/intermediate risk, CPX-351 for secondary AML.
  • Venetoclax + hypomethylating agent made unfit AML treatable, and since May 2026 the regimen can be fully oral.
  • Menin inhibitors (revumenib 2024/2025, ziftomenib 2025) opened NPM1-mutated and KMT2A-rearranged leukaemia, ~40% of adult AML, to a new drug class within one year.
  • MRD by flow and molecular methods now guides transplant, maintenance, and pre-emptive therapy; ELN 2021 MRD standards are in routine use.
  • Platform trials (myeloMATCH) assign therapy from rapid genomics at diagnosis and re-assign at each MRD checkpoint.
  • Allogeneic transplant is safer (post-transplant cyclophosphamide, haploidentical donors) and increasingly followed by targeted maintenance.
Who it affects
Show survival figures (1)

Averages across everyone diagnosed, often years ago. Your stage, subtype, age, fitness and the treatment you receive matter more than the average, and the numbers are improving quickly.

  • About 20,000 new cases a year in the US and 120,000 worldwide; median age 68; 5-year survival roughly 30% overall, above 60% in favourable-risk younger adults and below 10% in TP53-mutated disease.

Where the cases are

Cases by country · GLOBOCAN 2022
All countries →

Site: Leukaemia (all types) (shared total; subtype split not reported). World: 487,294 new cases, 305,405 deaths.

#CountryNew casesDeaths
1China81,94650,074
2United States of America63,14423,460
3India49,88336,871
4Germany15,1089,378
5Russian Federation14,4958,224
6Indonesia13,95910,370
7Japan13,57210,066
8France (metropolitan)13,5257,387
9Brazil11,8598,790
10Italy10,7997,197

GLOBOCAN reports leukaemia as one site; AML is roughly a quarter of cases worldwide.

Standard of care

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Fit

7+3 ± targeted agent; consolidation; allogeneic transplant by risk.

Relapsed

Genotype-directed: gilteritinib, IDH inhibitors, menin inhibitors; transplant.

Diagnosis and risk assignment

Marrow morphology, flow, karyotype/FISH, rapid FLT3/NPM1/IDH testing (results within days), NGS panel; ELN 2022 risk; fitness assessment. Menin-inhibitor and FLT3-inhibitor eligibility depends on these results.

Fit, FLT3-mutated

7+3 plus midostaurin (ITD or TKD) or quizartinib (ITD only), consolidation with continued inhibitor, allogeneic transplant for most FLT3-ITD in CR1, post-transplant FLT3-inhibitor maintenance if MRD-positive.

NCCN · Category 1 (midostaurin, quizartinib)ESMO-MCBS · A (RATIFY)
Fit, favourable or intermediate risk, CD33-positive

7+3 plus fractionated gemtuzumab ozogamicin (ALFA-0701); high-dose cytarabine consolidation; MRD-guided transplant for intermediate risk.

NCCN · Category 2A
Fit, secondary or therapy-related AML

CPX-351 induction (Study 301) then transplant in CR1; alternatives include 7+3 or venetoclax-based therapy in trials.

NCCN · Category 1 (age 60-75)
Fit, adverse risk (TP53, complex karyotype, MDS-related)

Intensive induction or venetoclax-azacitidine to remission, then allogeneic transplant as the only realistic cure; clinical trial strongly preferred; TP53-mutated disease has no effective targeted therapy after the magrolimab and eprenetapopt failures.

NCCN · Category 2A (clinical trial preferred)
Unfit for intensive chemotherapy (most patients over 75)

Venetoclax + azacitidine (VIALE-A) or venetoclax + oral decitabine-cedazuridine (ASCERTAIN-V, 2026); ivosidenib + azacitidine if IDH1-mutated (AGILE); low-dose cytarabine + venetoclax as an alternative. Continue until progression; consider transplant in responders who become fit.

NCCN · Category 1 (venetoclax + HMA)ESMO-MCBS · 4 (VIALE-A)
Maintenance after intensive therapy

Oral azacitidine (Onureg) for patients not transplanted (QUAZAR AML-001); FLT3 inhibitor maintenance after transplant in FLT3-ITD (MORPHO for MRD-positive); menin inhibitor maintenance in trials.

NCCN · Category 1 (oral azacitidine)
Relapsed or refractory, FLT3-mutated

Gilteritinib monotherapy (ADMIRAL) or gilteritinib + venetoclax/azacitidine, then transplant; quizartinib in Japan.

NCCN · Category 1
Relapsed or refractory, IDH-mutated

Ivosidenib or olutasidenib (IDH1), enasidenib (IDH2), often with azacitidine or venetoclax; differentiation-syndrome monitoring.

NCCN · Category 2A
Relapsed or refractory, NPM1-mutated or KMT2A-rearranged

Menin inhibitor: revumenib (KMT2Ar 2024; NPM1 2025) or ziftomenib (NPM1, November 2025), as a bridge to transplant; triplets with venetoclax-azacitidine in trials.

NCCN · Category 2A
Acute promyelocytic leukaemia

ATRA + arsenic trioxide without chemotherapy for standard risk (cure >95%); ATRA + arsenic + idarubicin or gemtuzumab for high risk. Differentiation syndrome prophylaxis.

NCCN · Category 1

Subtypes & biomarkers

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Subtypes
Biomarkers clinicians test
  • FLT3-ITD/TKD
  • NPM1
  • IDH1/2
  • KMT2A
  • TP53
  • CD33
  • ELN risk
  • MRD
  • ELN 2022 genetic risk group
  • FLT3-ITD and TKD (midostaurin, quizartinib, gilteritinib)
  • NPM1 (favourable risk without FLT3-ITD; MRD marker; menin inhibitor eligibility)
  • IDH1 / IDH2 (ivosidenib, olutasidenib, enasidenib)
  • KMT2A rearrangement (revumenib)
  • TP53 and complex karyotype (adverse; venetoclax less effective)
  • CD33 (gemtuzumab), CD123 (tagraxofusp, pivekimab)
  • Measurable residual disease (flow, NPM1 qPCR, NGS) after cycles 2 and before transplant
  • Karyotype/FISH at diagnosis
  • Myelodysplasia-related mutation set

Target prevalence in this cancer

Target / alterationPrevalenceSource
CD47
Magrolimab discontinued
>90%
Wikipedia
CD33
85-90%
Wikipedia
CD123
Universal in BPDCN
70-80%
Wikipedia
CD38
60-80%
Wikipedia
CD70
30-50%
Wikipedia
NPM1 mutation
~50-60% of cytogenetically normal AML
30%
FLT3
25-30%
cBioPortal (TCGA)
Menin
KMT2A rearrangement ~5-10%
25-30%
cBioPortal (TCGA)
IDH1 / IDH2
15-20%
cBioPortal (TCGA)
TP53
Higher in therapy-related AML
8-10%
cBioPortal (TCGA)
KMT2A (MLL) rearrangement
Higher in therapy-related AML
5-10%
BCL-2
n/a
Wikipedia

How common each drug target or alteration is in this cancer. Population-level and approximate; see the target page for detail. Full matrix.

History

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  1. 1948First chemotherapy remissions in leukaemia

    Farber's aminopterin in childhood ALL; AML remissions follow with 6-MP and cytarabine in the 1960s.

  2. 19737+3 regimen
  3. 19737+3 induction defined

    Cytarabine 7 days + daunorubicin 3 days (Yates et al.); still the intensive backbone.

  4. 1977First allogeneic transplants cure refractory leukaemia

    Thomas (Seattle) reports long-term survival after HLA-matched sibling transplant; Nobel Prize 1990.

  5. 1988ATRA induces differentiation in APL

    Shanghai group shows all-trans retinoic acid remissions; arsenic follows in the 1990s. First differentiation therapy.

  6. 2000Gemtuzumab: first ADC
  7. 2000Gemtuzumab ozogamicin, the first ADC

    Accelerated approval in relapsed CD33+ AML; withdrawn 2010 after SWOG S0106 toxicity.

  8. 2004Azacitidine approved (MDS)

    First hypomethylating agent; later the AML backbone for venetoclax and IDH/menin combinations.

  9. 2012ALFA-0701 rescues gemtuzumab

    Fractionated dosing with 7+3 improves EFS; re-approval 2017.

  10. 2017Midostaurin, enasidenib, gemtuzumab re-approval
  11. 2017Four approvals in one year

    Midostaurin (RATIFY), enasidenib, CPX-351, gemtuzumab re-approval; the first new AML drugs since 2000.

  12. 2018Ivosidenib, gilteritinib, and venetoclax combinations

    Ivosidenib (IDH1) and gilteritinib (ADMIRAL) approved; venetoclax + HMA/LDAC gets accelerated approval for unfit AML.

  13. 2020VIALE-A: venetoclax-azacitidine improves survival in unfit AML

    OS 14.7 vs 9.6 months; full approval October 2020; oral azacitidine maintenance approved (QUAZAR).

  14. 2022ELN 2022 risk, WHO/ICC classifications, AGILE, olutasidenib

    Genetics-first classification; ivosidenib-azacitidine OS HR 0.44; second IDH1 inhibitor approved.

  15. 2023Quizartinib approved in frontline FLT3-ITD AML

    QuANTUM-First OS 31.9 vs 15.1 months, including patients to age 75.

  16. 2024Revumenib: first menin inhibitor
  17. 2024Revumenib: first menin inhibitor; magrolimab fails

    Approved for KMT2A-rearranged acute leukaemia (AUGMENT-101). Magrolimab (CD47) discontinued after ENHANCE trials, a setback for TP53-mutated AML.

  18. 2025Menin inhibitors reach NPM1-mutated AML

    Revumenib NPM1 label (October) and ziftomenib approval (13 November, KOMET-001).

  19. 2026First all-oral AML regimen

    Decitabine-cedazuridine + venetoclax approved 13 May 2026 (ASCERTAIN-V, CR 41.6%).

Pipeline

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Open problems

  • TP53-mutant AML remains lethal.
  • Older patients.
  • TP53-mutated and complex-karyotype AML: no class has improved survival; magrolimab (CD47) and eprenetapopt (p53 reactivator) both failed in phase 3.
  • Relapse after allogeneic transplant remains the leading cause of death; which maintenance (FLT3, menin, azacitidine) helps whom is unresolved.
  • Menin-inhibitor resistance through MEN1 mutations appears within months in a third of relapsing patients; combinations and next-generation inhibitors are needed.
  • Early death from infection and cytopenias on venetoclax-based therapy in the very old; optimal venetoclax duration is untested in randomised trials.
  • MRD thresholds and assays are not harmonised across labs, and CHIP-associated mutations confound NGS MRD.
  • Whether triplets (menin or FLT3 inhibitor + venetoclax + HMA) improve survival over doublets, and at what toxicity, awaits phase 3.
  • Access: rapid genomics within 72 hours and menin/FLT3 inhibitors are unavailable in most low- and middle-income settings.

Trials

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Recruiting now (live from ClinicalTrials.gov)

Recruiting trials near you · live from ClinicalTrials.gov
Acute myeloid leukaemia
condition: acute myeloid leukemia
Open on ClinicalTrials.gov →

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Landmark trials in OnCo

Expert centres

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Where the expertise is

Centres linked to this cancer in OnCo

Seeking a second opinion: ask your oncologist for a referral to a high-volume centre; most accept records and pathology by mail or telehealth. In the US, use the NCI's Find a Cancer Center tool or the nonprofit Cancer Commons, which navigates options for advanced cancers at no cost.

Questions to ask

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Bring to your appointment

Questions to ask your oncologist about Acute myeloid leukaemia

Generated from this cancer's standard of care, biomarkers, and pipeline · 41 questions

Newly diagnosed

  1. What is my exact diagnosis, stage, and grade, and which tests established them?
    Why: Everything else follows from an accurate stage and subtype.
  2. Which biomarkers have been tested on my tumour (for example FLT3-ITD/TKD, NPM1, IDH1/2, KMT2A, TP53), and what were the results?
    Why: These results decide eligibility for targeted therapy, immunotherapy, and trials.
  3. Which subtype is my cancer, and does that change the recommended treatment?
    Why: Recognised subtypes for this cancer include AML with defining genetic abnormalities: NPM1-mutated, CEBPA bZIP, RUNX1::RUNX1T1, CBFB::MYH11, KMT2A-rearranged, DEK::NUP214, BCR::ABL1, MECOM, Acute promyelocytic leukaemia, curable without chemotherapy in most cases, AML, myelodysplasia-related.
  4. Is germline (inherited) genetic testing recommended for me or my family?
    Why: Inherited variants can change treatment and matter for relatives.

Fit

  1. For my situation (fit), which of the standard options do you recommend and why?
    Why: Guideline options include: 7+3 ± targeted agent; consolidation; allogeneic transplant by risk.
  2. Am I a candidate for Gemtuzumab ozogamicin, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.

Unfit

  1. For my situation (unfit), which of the standard options do you recommend and why?
    Why: Guideline options include: Azacitidine + venetoclax.
  2. Am I a candidate for Venetoclax, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.

Relapsed

  1. For my situation (relapsed), which of the standard options do you recommend and why?
    Why: Guideline options include: Genotype-directed: gilteritinib, IDH inhibitors, menin inhibitors; transplant.
  2. Am I a candidate for Revumenib, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.

Diagnosis and risk assignment

  1. For my situation (diagnosis and risk assignment), which of the standard options do you recommend and why?
    Why: Guideline options include: Marrow morphology, flow, karyotype/FISH, rapid FLT3/NPM1/IDH testing (results within days), NGS panel; ELN 2022 risk; fitness assessment. Menin-inhibitor and FLT3-inhibitor eligibility depends on these results.

Fit, FLT3-mutated

  1. For my situation (fit, flt3-mutated), which of the standard options do you recommend and why?
    Why: Guideline options include: 7+3 plus midostaurin (ITD or TKD) or quizartinib (ITD only), consolidation with continued inhibitor, allogeneic transplant for most FLT3-ITD in CR1, post-transplant FLT3-inhibitor maintenance if MRD-positive.
  2. Am I a candidate for Cytarabine + anthracycline ('7+3'), Midostaurin, Quizartinib, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.
  3. How do the results of RATIFY (CALGB 10603) and QuANTUM-First apply to someone like me?
    Why: Trial populations differ from individual patients; ask how closely you match.

Fit, favourable or intermediate risk, CD33-positive

  1. For my situation (fit, favourable or intermediate risk, cd33-positive), which of the standard options do you recommend and why?
    Why: Guideline options include: 7+3 plus fractionated gemtuzumab ozogamicin (ALFA-0701); high-dose cytarabine consolidation; MRD-guided transplant for intermediate risk.
  2. Am I a candidate for Gemtuzumab ozogamicin, Cytarabine + anthracycline ('7+3'), and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.
  3. How do the results of ALFA-0701 apply to someone like me?
    Why: Trial populations differ from individual patients; ask how closely you match.

Fit, secondary or therapy-related AML

  1. For my situation (fit, secondary or therapy-related aml), which of the standard options do you recommend and why?
    Why: Guideline options include: CPX-351 induction (Study 301) then transplant in CR1; alternatives include 7+3 or venetoclax-based therapy in trials.
  2. Am I a candidate for CPX-351 (liposomal daunorubicin-cytarabine), and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.
  3. How do the results of CPX-351 Study 301 apply to someone like me?
    Why: Trial populations differ from individual patients; ask how closely you match.

Fit, adverse risk (TP53, complex karyotype, MDS-related)

  1. For my situation (fit, adverse risk (tp53, complex karyotype, mds-related)), which of the standard options do you recommend and why?
    Why: Guideline options include: Intensive induction or venetoclax-azacitidine to remission, then allogeneic transplant as the only realistic cure; clinical trial strongly preferred; TP53-mutated disease has no effective targeted therapy after the magrolimab and eprenetapopt failures.
  2. Am I a candidate for Venetoclax, Azacitidine, Magrolimab, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.

Unfit for intensive chemotherapy (most patients over 75)

  1. For my situation (unfit for intensive chemotherapy (most patients over 75)), which of the standard options do you recommend and why?
    Why: Guideline options include: Venetoclax + azacitidine (VIALE-A) or venetoclax + oral decitabine-cedazuridine (ASCERTAIN-V, 2026); ivosidenib + azacitidine if IDH1-mutated (AGILE); low-dose cytarabine + venetoclax as an alternative. Continue until progression; consider transplant in responders who become fit.
  2. Am I a candidate for Venetoclax, Azacitidine, Decitabine + cedazuridine (oral) or related drugs, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.
  3. How do the results of VIALE-A and AGILE apply to someone like me?
    Why: Trial populations differ from individual patients; ask how closely you match.

Maintenance after intensive therapy

  1. For my situation (maintenance after intensive therapy), which of the standard options do you recommend and why?
    Why: Guideline options include: Oral azacitidine (Onureg) for patients not transplanted (QUAZAR AML-001); FLT3 inhibitor maintenance after transplant in FLT3-ITD (MORPHO for MRD-positive); menin inhibitor maintenance in trials.
  2. Am I a candidate for Azacitidine, Gilteritinib, Quizartinib, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.

Relapsed or refractory, FLT3-mutated

  1. For my situation (relapsed or refractory, flt3-mutated), which of the standard options do you recommend and why?
    Why: Guideline options include: Gilteritinib monotherapy (ADMIRAL) or gilteritinib + venetoclax/azacitidine, then transplant; quizartinib in Japan.
  2. Am I a candidate for Gilteritinib, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.
  3. How do the results of ADMIRAL apply to someone like me?
    Why: Trial populations differ from individual patients; ask how closely you match.

Relapsed or refractory, IDH-mutated

  1. For my situation (relapsed or refractory, idh-mutated), which of the standard options do you recommend and why?
    Why: Guideline options include: Ivosidenib or olutasidenib (IDH1), enasidenib (IDH2), often with azacitidine or venetoclax; differentiation-syndrome monitoring.
  2. Am I a candidate for Ivosidenib, Olutasidenib, Enasidenib, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.

Relapsed or refractory, NPM1-mutated or KMT2A-rearranged

  1. For my situation (relapsed or refractory, npm1-mutated or kmt2a-rearranged), which of the standard options do you recommend and why?
    Why: Guideline options include: Menin inhibitor: revumenib (KMT2Ar 2024; NPM1 2025) or ziftomenib (NPM1, November 2025), as a bridge to transplant; triplets with venetoclax-azacitidine in trials.
  2. Am I a candidate for Revumenib, Ziftomenib, and what side effects should I expect?
    Why: Knowing the expected toxicities helps you plan work, family, and supportive care.
  3. How do the results of AUGMENT-101 and KOMET-001 apply to someone like me?
    Why: Trial populations differ from individual patients; ask how closely you match.

Acute promyelocytic leukaemia

  1. For my situation (acute promyelocytic leukaemia), which of the standard options do you recommend and why?
    Why: Guideline options include: ATRA + arsenic trioxide without chemotherapy for standard risk (cure >95%); ATRA + arsenic + idarubicin or gemtuzumab for high risk. Differentiation syndrome prophylaxis.

Any stage

  1. Are there clinical trials I could join, for example of Revumenib, Venetoclax, Ziftomenib, Menin inhibitor + venetoclax + azacitidine?
    Why: Trials are how the next standard of care is set; asking early keeps options open.
  2. Would a second opinion at a high-volume centre change anything, and can you help arrange it?
    Why: Rare or high-stakes decisions benefit from a centre that treats many similar patients.
  3. What supportive care (symptom control, nutrition, exercise, mental health, financial help) is available from the start?
    Why: Supportive care improves quality of life and helps patients complete treatment.
  4. I read that “TP53-mutant AML remains lethal”. How does that affect my plan?
    Why: Open problems are where trials and second opinions matter most.
  5. I read that “Older patients”. How does that affect my plan?
    Why: Open problems are where trials and second opinions matter most.

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Everything relevant

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Direct links plus the targets, companies, and technologies of this cancer's products.

technologies

15

targets

17

drugs

24
Not mapped hereInorganic arsenical (differentiation agent)
Arsenic trioxide · Trisenox
ApprovedSmall-molecule hypomethylating agent (cytotoxic)
Azacitidine · Vidaza / Onureg (oral)
Not mapped hereOral ROCK2 inhibitor
Belumosudil · Rezurock
ApprovedLiposomal cytotoxic formulation
CPX-351 (liposomal daunorubicin-cytarabine) · Vyxeos
Not mapped hereCytotoxic regimen
Cytarabine + anthracycline ('7+3')
ApprovedOral hypomethylating agent
Decitabine + cedazuridine (oral) · Inqovi
ApprovedSmall-molecule IDH2 inhibitor
Enasidenib · Idhifa
NegativeSmall molecule (p53 reactivator)
Eprenetapopt
Not mapped hereTopoisomerase II inhibitor (podophyllotoxin derivative)
Etoposide · VePesid / Etopophos / Toposar
ApprovedADC
Gemtuzumab ozogamicin · Mylotarg
ApprovedSmall-molecule kinase inhibitor (FLT3, type I)
Gilteritinib · Xospata
Not mapped hereSmall-molecule smoothened (hedgehog) inhibitor
Glasdegib · Daurismo
ApprovedSmall-molecule IDH1 inhibitor
Ivosidenib · Tibsovo
WithdrawnMonoclonal antibody (anti-CD47)
Magrolimab
ApprovedSmall-molecule multikinase inhibitor (FLT3)
Midostaurin · Rydapt
ApprovedSmall-molecule IDH1 inhibitor
Olutasidenib · Rezlidhia
Not mapped hereADC (anti-CD123 antibody, IGN payload)
Pivekimab sunirine · Decnupaz
ApprovedSmall-molecule kinase inhibitor (FLT3-ITD, type II)
Quizartinib · Vanflyta
ApprovedSmall-molecule menin inhibitor
Revumenib · Revuforj
ApprovedRecombinant cytotoxin (IL-3 fused to diphtheria toxin)
Tagraxofusp · Elzonris
Not mapped hereAlkylating conditioning agent (busulfan analogue)
Treosulfan · Grafapex
Not mapped hereOral retinoid (differentiation agent)
Tretinoin (all-trans retinoic acid, ATRA) · Vesanoid
ApprovedSmall-molecule BCL-2 inhibitor
Venetoclax · Venclexta
ApprovedSmall-molecule menin inhibitor
Ziftomenib · Komzifti

companies

17

institutions

47
American Society of HematologyAuckland City Hospital / Te Pūriri o Te Ora Cancer and Blood ServiceCancer Research UK Manchester InstituteChao Family Comprehensive Cancer Center, UC IrvineChildren's Cancer Hospital Egypt 57357Chinese PLA General HospitalChristian Medical College, VelloreComprehensive Cancer Center Freiburg (CCCF)Comprehensive Cancer Center Mainfranken, University Hospital WürzburgComprehensive Cancer Center Tübingen-StuttgartEuropean Hematology AssociationGIMEMAGreat Ormond Street Hospital for ChildrenHamad Medical Corporation / National Center for Cancer Care and ResearchHospital Universitari i Politècnic La FeHospital Universitario 12 de OctubreHOVONHUS Comprehensive Cancer Center, Helsinki University HospitalInstitut Paoli-CalmettesIRCCS Azienda Ospedaliero-Universitaria di Bologna – Policlinico Sant'OrsolaIRCCS Ospedale San RaffaeleKyoto University HospitalMasonic Cancer Center, University of MinnesotaMontefiore Einstein Comprehensive Cancer CenterNational Taiwan University HospitalNational University Hospital / National University Cancer Institute, SingaporeNCT/UCC Dresden – University Hospital Carl Gustav CarusOHSU Knight Cancer InstituteOxford Cancer – Oxford University Hospitals and University of OxfordPrincess Máxima Center for Pediatric OncologyQueen Mary Hospital / University of Hong KongRamathibodi Hospital, Mahidol UniversityRambam Health Care CampusRigshospitalet – Copenhagen University HospitalRoyal Adelaide HospitalRuijin Hospital, Shanghai Jiao Tong UniversitySeoul St. Mary's HospitalSiriraj Hospital, Mahidol UniversitySylvester Comprehensive Cancer Center, University of MiamiTata Medical Center, KolkataThe Ohio State University Comprehensive Cancer Center – James Cancer Hospital and Solove Research InstituteUniversity Cancer Center Frankfurt (UCT)USC Norris Comprehensive Cancer CenterVCU Massey Comprehensive Cancer CenterWalter and Eliza Hall Institute of Medical ResearchWeizmann Institute of ScienceWest German Cancer Center (WTZ), University Hospital Essen

pathways

4

terms

6

trials

11

pairings

3

ideas

7

collections

1

people

24

bottlenecks

4

key papers

6

Key papers

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translationalNature 2023changed practice
AUGMENT-101: revumenib, the first menin inhibitor, in relapsed leukaemias driven by KMT2A rearrangement or NPM1 mutation

Revumenib proved that a transcriptional dependency, rather than a kinase, can be drugged in leukaemia, opening treatment for two genetic subgroups that together cover roughly a third of AML plus most infant ALL. It is now approved and is being combined with venetoclax-azacitidine and intensive chemotherapy in front-line trials. Single-agent remissions are often short without transplant.

rctThe Lancet 2023changed practice
QuANTUM-First: quizartinib added to intensive chemotherapy and continued as maintenance in newly diagnosed FLT3-ITD AML

QuANTUM-First gave FLT3-ITD AML patients a second front-line targeted option and showed that continuing a FLT3 inhibitor as long-term maintenance, including after transplant, pays off. Quizartinib was approved for this indication in 2023. Head-to-head data against midostaurin are lacking, and the design leaves open how much of the benefit came from maintenance.

rctNew England Journal of Medicine 2022changed practice
AGILE: ivosidenib plus azacitidine for newly diagnosed IDH1-mutated AML in patients unfit for intensive chemotherapy

AGILE showed that for the roughly 6-10% of AML patients with an IDH1 mutation, a targeted doublet produces survival in the range of two years, an outcome previously unimaginable in unfit patients. Ivosidenib-azacitidine is approved and is one option alongside venetoclax-azacitidine for these patients. Which regimen, or triplet, is best for IDH1-mutated disease has not been settled by a randomised trial.

rctNew England Journal of Medicine 2020changed practice
VIALE-A: venetoclax plus azacitidine for older adults with acute myeloid leukaemia who cannot have intensive chemotherapy

VIALE-A turned a palliative regimen into one that produces remission in two-thirds of older AML patients and is now the reference treatment for anyone not fit for intensive chemotherapy. It shifted the field towards lower-intensity targeted combinations and opened the door to adding FLT3, IDH and menin inhibitors to the backbone. Cure remains uncommon and most patients relapse within two years.

rctNew England Journal of Medicine 2019changed practice
ADMIRAL: gilteritinib pills versus chemotherapy for relapsed FLT3-mutated acute myeloid leukaemia

ADMIRAL showed that a targeted oral drug can beat chemotherapy outright in relapsed AML, and made gilteritinib the standard bridge to transplant for FLT3-mutated relapse. Its success also underpinned FLT3 inhibitor use in first-line combinations. Resistance through FLT3-independent clones and RAS pathway mutations limits durability without transplant.

observationalNew England Journal of Medicine 2014
Jaiswal: clonal haematopoiesis, the pre-leukaemic clones in most people over 70

Many older people carry blood clones one or two steps from leukaemia, and those clones also drive heart disease through inflammation. CHIP is why blood-based cancer tests must filter out mutations from blood cells, and it opens a route to preventing both leukaemia and cardiovascular events in carriers.

Latest papers

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Query for this cancer: (TITLE:"Acute myeloid leukaemia" OR ABSTRACT:"Acute myeloid leukaemia") AND (treatment OR therapy OR trial OR survival OR diagnosis). Results are unfiltered search hits about Acute myeloid leukaemia, not a curated reading list.

Connected

177top

technologies

12

targets

16

drugs

24
Not mapped hereInorganic arsenical (differentiation agent)
Arsenic trioxide · Trisenox
ApprovedSmall-molecule hypomethylating agent (cytotoxic)
Azacitidine · Vidaza / Onureg (oral)
Not mapped hereOral ROCK2 inhibitor
Belumosudil · Rezurock
ApprovedLiposomal cytotoxic formulation
CPX-351 (liposomal daunorubicin-cytarabine) · Vyxeos
Not mapped hereCytotoxic regimen
Cytarabine + anthracycline ('7+3')
ApprovedOral hypomethylating agent
Decitabine + cedazuridine (oral) · Inqovi
ApprovedSmall-molecule IDH2 inhibitor
Enasidenib · Idhifa
NegativeSmall molecule (p53 reactivator)
Eprenetapopt
Not mapped hereTopoisomerase II inhibitor (podophyllotoxin derivative)
Etoposide · VePesid / Etopophos / Toposar
ApprovedADC
Gemtuzumab ozogamicin · Mylotarg
ApprovedSmall-molecule kinase inhibitor (FLT3, type I)
Gilteritinib · Xospata
Not mapped hereSmall-molecule smoothened (hedgehog) inhibitor
Glasdegib · Daurismo
ApprovedSmall-molecule IDH1 inhibitor
Ivosidenib · Tibsovo
WithdrawnMonoclonal antibody (anti-CD47)
Magrolimab
ApprovedSmall-molecule multikinase inhibitor (FLT3)
Midostaurin · Rydapt
ApprovedSmall-molecule IDH1 inhibitor
Olutasidenib · Rezlidhia
Not mapped hereADC (anti-CD123 antibody, IGN payload)
Pivekimab sunirine · Decnupaz
ApprovedSmall-molecule kinase inhibitor (FLT3-ITD, type II)
Quizartinib · Vanflyta
ApprovedSmall-molecule menin inhibitor
Revumenib · Revuforj
ApprovedRecombinant cytotoxin (IL-3 fused to diphtheria toxin)
Tagraxofusp · Elzonris
Not mapped hereAlkylating conditioning agent (busulfan analogue)
Treosulfan · Grafapex
Not mapped hereOral retinoid (differentiation agent)
Tretinoin (all-trans retinoic acid, ATRA) · Vesanoid
ApprovedSmall-molecule BCL-2 inhibitor
Venetoclax · Venclexta
ApprovedSmall-molecule menin inhibitor
Ziftomenib · Komzifti

companies

12

institutions

47
American Society of HematologyAuckland City Hospital / Te Pūriri o Te Ora Cancer and Blood ServiceCancer Research UK Manchester InstituteChao Family Comprehensive Cancer Center, UC IrvineChildren's Cancer Hospital Egypt 57357Chinese PLA General HospitalChristian Medical College, VelloreComprehensive Cancer Center Freiburg (CCCF)Comprehensive Cancer Center Mainfranken, University Hospital WürzburgComprehensive Cancer Center Tübingen-StuttgartEuropean Hematology AssociationGIMEMAGreat Ormond Street Hospital for ChildrenHamad Medical Corporation / National Center for Cancer Care and ResearchHospital Universitari i Politècnic La FeHospital Universitario 12 de OctubreHOVONHUS Comprehensive Cancer Center, Helsinki University HospitalInstitut Paoli-CalmettesIRCCS Azienda Ospedaliero-Universitaria di Bologna – Policlinico Sant'OrsolaIRCCS Ospedale San RaffaeleKyoto University HospitalMasonic Cancer Center, University of MinnesotaMontefiore Einstein Comprehensive Cancer CenterNational Taiwan University HospitalNational University Hospital / National University Cancer Institute, SingaporeNCT/UCC Dresden – University Hospital Carl Gustav CarusOHSU Knight Cancer InstituteOxford Cancer – Oxford University Hospitals and University of OxfordPrincess Máxima Center for Pediatric OncologyQueen Mary Hospital / University of Hong KongRamathibodi Hospital, Mahidol UniversityRambam Health Care CampusRigshospitalet – Copenhagen University HospitalRoyal Adelaide HospitalRuijin Hospital, Shanghai Jiao Tong UniversitySeoul St. Mary's HospitalSiriraj Hospital, Mahidol UniversitySylvester Comprehensive Cancer Center, University of MiamiTata Medical Center, KolkataThe Ohio State University Comprehensive Cancer Center – James Cancer Hospital and Solove Research InstituteUniversity Cancer Center Frankfurt (UCT)USC Norris Comprehensive Cancer CenterVCU Massey Comprehensive Cancer CenterWalter and Eliza Hall Institute of Medical ResearchWeizmann Institute of ScienceWest German Cancer Center (WTZ), University Hospital Essen

pathways

4

terms

6

trials

11

pairings

3

ideas

7

collections

1

people

24

bottlenecks

4

key papers

6